Phosphodiesterases as Drug Targets

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431,95 
Įprasta kaina: 508,18 
-15% su kodu: ENG15
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Akcija baigiasi: 2025-03-03
-15% su kodu: ENG15
431,95 
Įprasta kaina: 508,18 
-15% su kodu: ENG15
Kupono kodas: ENG15
Akcija baigiasi: 2025-03-03
-15% su kodu: ENG15
2025-02-28 508.1800 InStock
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Knygos aprašymas

Cyclic nucleotide phosphodiesterases (PDEs) are promising targets for pharmacological intervention. Multiple PDE genes, isoform diversity, selective expression and compartmentation of the isoforms, and an array of conformations of PDE proteins are properties that challenge development of drugs that selectively target this class of enzymes. Novel characteristics of PDEs are viewed as unique opportunities to increase specificity and selectivity when designing novel compounds for certain therapeutic indications. This chapter provides a summary of the major concepts related to the design and use of PDE inhibitors.

Informacija

Serija: Handbook of Experimental Pharmacology
Leidėjas: Springer Berlin Heidelberg
Išleidimo metai: 2013
Knygos puslapių skaičius: 540
ISBN-10: 3642269451
ISBN-13: 9783642269455
Formatas: 235 x 155 x 29 mm. Knyga minkštu viršeliu
Kalba: Anglų

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